Active Ingredient History

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Thiocolchicoside is a muscle relaxant with anti-inflammatory and analgesic effects. How it works is unknown, but it is believed to be via antagonism of nicotinic acetylcholine receptors. However, it is also appears to be a competitive antagonist of GABAA and glycine receptors. As such, it has powerful convulsant activity and should not be used in seizure-prone individuals.   Wikipedia

  • SMILES: COc1c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)cc3CCC(NC(=O)C)C4=CC(=O)C(=CC=C4c3c1OC)SC
  • InChIKey: LEQAKWQJCITZNK-MSQQGMGVSA-N
  • Mol. Mass: 563.63
  • ALogP: 0.76
  • ChEMBL Molecule:
More Chemistry
2,14-di-(demethoxy)-2-glucosidoxy-14- methylthiocolchicine | coltramyl | miorel | muscoril | myoplège | thiocholshikoside | thiocolchicine 2-glucoside analog | thiocolchicine glycoside | thiocolchicoside

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