Active Ingredient History

  • Now
Eletriptan (eletriptan hydrobromide, trade name Relpax) is a selective 5-hydroxytryptamine (5-HT1B/1D) serotonin receptor agonist (triptan) indicated for the acute treatment of migraine with or without aura in adults. Eletriptan binds with high affinity to 5-HT1B, 5-HT1D and 5-HT1F receptors, and has modest affinity for 5-HT1A, 5-HT1E, 5-HT2B and 5-HT7 receptors. The therapeutic activity of eletriptan for the treatment of migraine headache is thought to be due to the agonist effects at the 5-HT1B/1D receptors on intracranial blood vessels (including the arterio-venous anastomoses) and sensory nerves of the trigeminal system which result in cranial vessel constriction and inhibition of pro-inflammatory neuropeptide release. Eletriptan (Relpax) has been approved for use in the acute treatment of migraine in 51 countries and has been introduced in 17 countries including Mexico, Italy, France and Japan.   NCATS

  • SMILES: CN1CCC[C@@H]1Cc2c[nH]c3ccc(CCS(=O)(=O)c4ccccc4)cc23
  • Mol. Mass: 382.53
  • ALogP: 3.82
  • ChEMBL Molecules:
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Drug Pricing (per unit)

United States

$0.1033 - $100.0700
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Note: This drug pricing data is preliminary, incomplete, and may contain errors.

3-(1-methyl-2-pyrrolidinylmethyl)-5-(2-(phenylsulfonyl)ethyl)-1h-indole hydrobromide | eletriptan | eletriptan hydrobromide | eletriptanum | (r)-3-((1-methyl-2-pyrrolidinyl)methyl)-5-(2-(phenylsulfonyl)ethyl)-1h-indole | (r)-3-((1-methyl-2-pyrrolidinyl)methyl)-5-(2-(phenylsulfonyl)ethyl)-1h-indole monohydrobromide | relpax | uk-116044 | uk-116,044 | uk 116044-04 | uk-11604404 | uk-116,044-04 | uk-116044-04 | uk-116044-04 [as hydrobromide) | uk 166044 | uk 166,044 | uk-166044 | uk-166,044


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