apitolisib Report issue

Small molecule Experimental
AACT ChEMBL DrugBank MeSH PubChem

Active Ingredient History

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Chemistry

  • SMILES: C[C@H](O)C(=O)N1CCN(Cc2sc3c(nc(nc3c2C)c4cnc(N)nc4)N5CCOCC5)CC1
  • InChIKey: YOVVNQKCSKSHKT-HNNXBMFYSA-N
  • Mol. Mass: 498.61
  • ALogP: 0.9
  • ChEMBL Molecule:
    apitolisib  
More Chemistry

Pharmacology

Alternative names

1-(4-((2-(2-aminopyrimidin-5-yl)-7-methyl-4-morpholinothieno(3,2-d)pyrimidin-6-yl)methyl)piperazin-1-yl)-2-hydroxypropan-1-one | apitolisib | g-038390 | g-038390.1 | gdc0980 | gdc 0980 | gdc-0980 | gdc-0980.1 | rg-7422

Organizations (1)

Research & Development (1)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Marketing (0)

Organization Org Type FDA approvals Clinical Trials involvement Org ID Force Sort

Indications (7)

Approved Indications (0)

Experimental Indications - Clinical Trial Phases 1-4 (7)


 

Breast Neoplasms (Phase 2)

Carcinoma, Renal Cell (Phase 2)

Endometrial Neoplasms (Phase 2)

Healthy Volunteers (Phase 1)

Lymphoma, Non-Hodgkin (Phase 1)

Neoplasms (Phase 1)

Prostatic Neoplasms (Phase 1/Phase 2)

Overview

  • Highest Phase: Phase 2
  • # of Trials: 12
  • # of Trial Organizations: 1

Trials by Phase

Trial Phase Start Date Organizations Indications

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