Active Ingredient History

  • Now
Nabilone is a synthetic cannabinoid approved under the brand name cesamet for treatment of severe nausea and vomiting associated with cancer chemotherapy. Nabilone is an orally active which, like other cannabinoids, has complex effects on the central nervous system (CNS). It has been suggested that the antiemetic effect of nabilone is caused by interaction with the cannabinoid receptor system, i.e. the CB (1) receptor, which has been discovered in neural tissues.   NCATS

  • SMILES: CCCCCCC(C)(C)C1=CC(O)=C2[C@@H]3CC(=O)CC[C@H]3C(C)(C)OC2=C1
  • Mol. Mass: 372.5408
  • ALogP: 6.26
  • ChEMBL Molecules:
More Chemistry
  • Mechanism of Action:
  • Multi-specific: Missing data
  • Black Box: No
  • Availability: Prescription Only
  • Delivery Methods: Oral
  • Pro Drug: No
3-(1,1-dimethylheptyl)-6,6a,7,8,10,10a- hexahydro-1-hydroxy-6,6-dimethyl-9h-dibenzo(b,d)pyran-9-one | cesamet | cesemat | cpd 109514 | cpd-109514 | lilly 109514 | lilly brand of nabilone | ly 109514 | ly-109514 | nabilon | nabilona | nabilone | nabilone, (6ar-trans)-isomer | nabilone, (6as-trans)-isomer | nabilone, (cis-(+-))-isomer | nabilone, (trans-(+-))-isomer | nabilonum


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